An efficient protocol for the solid-phase synthesis of malondiamides.

نویسندگان

  • Markus M Vögtle
  • Andreas L Marzinzik
چکیده

A novel and straightforward solid-phase synthesis of malondiamides containing a free nitrogen has been developed. These intermediates, which can be directly obtained in good yield and purity, can be further derivatised. This approach can be used for the synthesis of large split-and-mix-libraries.

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عنوان ژورنال:
  • Molecules

دوره 10 12  شماره 

صفحات  -

تاریخ انتشار 2005